Taking the time to study competitive antagonism

D. J. Wyllie, P. E. Chen

Research output: Contribution to journalArticlepeer-review

Original languageEnglish
Pages (from-to)541-51
Number of pages11
JournalBritish Journal of Pharmacology
Volume150
Issue number5
Publication statusPublished - 2007

Keywords

  • Animals *Binding, Competitive Computer Simulation Dose-Response Relationship, Drug Drug Evaluation, Preclinical/methods Excitatory Amino Acid Agonists/metabolism/pharmacology Excitatory Amino Acid Antagonists/metabolism/pharmacology Humans Ion Channel Gating/*drug effects Ion Channels/agonists/*antagonists & inhibitors/genetics/metabolism Kinetics *Ligands Models, Biological Nicotinic Agonists/metabolism/pharmacology Nicotinic Antagonists/metabolism/pharmacology Point Mutation Protein Binding Receptors, Cell Surface/agonists/*antagonists & inhibitors/genetics/metabolism Receptors, N-Methyl-D-Aspartate/antagonists & inhibitors Receptors, Nicotinic/drug effects Reproducibility of Results Synaptic Transmission/drug effects

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